Bioanalytical Community

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  • 1.  Immunoaffinity LC-MS for measuring protein therapeutics and biomarkers

    Community Leadership
    Posted 07-31-2023 13:41

    During the recent monthly PK assay working group meeting, Dr. Keyang Xu from Genentech/Roche presented valuable insights into the strategy and practices of utilizing Immunoaffinity LC-MS for measuring protein therapeutics and biomarkers. The following key take-home messages were highlighted:

    • Immunoaffinity capture LC-MS offers a reliable and effective alternative to LBA (ligand-binding assays) in the bioanalysis of protein drugs and targets.
    • Understanding which analyte(s) to measure is crucial, considering factors such as the impact of biotransformation on the results.
    • Bioanalytical assay strategies can encompass both generic and specific approaches, catering to the unique requirements of the study.
    • Starting with LBA acceptance criteria is recommended as a solid foundation for assay development, validation, and sample analysis.

    The monthly PK Assay Working Group gathering, focusing on PK Methodologies for Biologics, Cell, and Gene therapies, provides an invaluable platform for industry experts to come together. During these meetings, we collaboratively share best practices, tackle emerging challenges, and exchange valuable experiences. The primary goal is to support each other in refining PK methodologies and facilitating successful filling and submission processes.



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    Mark Ma, Ph.D.
    Head of Translational Clinical Sciences
    Rallybio
    New Haven CT
    [email protected]

    Disclaimer: Opinions expressed are solely my own and do not express the views or opinions of my employer.
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  • 2.  RE: Immunoaffinity LC-MS for measuring protein therapeutics and biomarkers

    Community Leadership
    Posted 08-07-2023 17:35

    Great topic! One point I like to emphasize is the value of adding a true internal standard that can capture impact of all processing steps. This is particularly important when considering the impact of potential interfering substances such as target and anti-drug antibodies. A peptide alone will not capture this. Fortunately, I have seen increased emphasis on the use of appropriate internal standards in recent AAPS work.



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    Joleen White Ph.D.
    AAPS 2023 Global Health Community Past Chair
    Bioanalytical 101 Course Development
    Head of Bioassay Development
    Gates Medical Research Institute
    Cambridge MA
    [email protected]

    Disclaimer: Opinions expressed are solely my own and do not express the views or opinions of my employer.
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  • 3.  RE: Immunoaffinity LC-MS for measuring protein therapeutics and biomarkers

    Posted 08-08-2023 11:13

    Thanks Mark for the update and leading this important topic. IA-LC-MS/MS is and will become more popular as biologics/biomarkers drive therapeutics. MS/MS is now sensitive enough to capture many of the LLOQs that weren't achievable by LC-MS/MS even a decade ago. That powered with the additional selectivity of a immuno assay clean-up (on-line or off-line) gives the best of both worlds. I also like to see now we have some general approaches for IA before LC-MS/MS, so we can take method development to days/weeks instead of months....



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    Shane Needham
    Founder, President and CEO
    Veloxity Labs, LLC
    Peoria IL
    [email protected]

    Disclaimer: Opinions expressed are solely my own and do not express the views or opinions of my employer.
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  • 4.  RE: Immunoaffinity LC-MS for measuring protein therapeutics and biomarkers

    Community Leadership
    Posted 08-10-2023 12:15

    This is great information!  Thanks Mark!  



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    Jim Shen PhD
    Executive Director, Head of Regulated Bioanalysis Operations
    Bristol-Myers Squibb
    Princeton NJ
    [email protected]

    Disclaimer: Opinions expressed are solely my own and do not express the views or opinions of my employer.
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