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FDA Final Guidance: Clinical Pharmacology Considerations for Human Radiolabeled Mass Balance Studies

  • 1.  FDA Final Guidance: Clinical Pharmacology Considerations for Human Radiolabeled Mass Balance Studies

    Posted 07-22-2024 08:03

    This FDA Guidance has a narrow scope as described in the Introduction:

    "This guidance describes the FDA's recommendations regarding clinical pharmacology
    considerations for conducting human radiolabeled mass balance studies of investigational drugs,
    including: (1) deciding whether and when to conduct the study, (2) designing the study, and (3)
    reporting results.2 The recommendations in this guidance are, in part, based on the FDA's
    experience reviewing human radiolabeled mass balance studies submitted to the Agency in
    recent new drug applications (NDAs).3 This guidance does not cover animal mass balance
    studies, safety testing of drug metabolites, or recommendations for selecting the radioactivity
    dose."

    In the Background section, a succinct statement on why radiolabeled mass balance studies are conducted:

    "A human radiolabeled (most commonly 14C or 3H) mass balance study is the single most direct method to obtain quantitative and comprehensive information on the absorption, distribution, metabolism, and excretion (ADME) of the drug in the human body."

    #fda  #massbalance  #radiolabeled #Guidance

    Clin Pharm Considerations for Human Radiolabeled Mass Balance Studies

    U.S. Food and Drug Administration remove preview


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    Mark Arnold Ph.D., FAAPS
    Westampton, NJ
    [email protected]
    Bioanalytical Solution Integration
    LinkedIn: https://www.linkedin.com/in/markearnoldphd/
    Website & Blog: Bioanalysis & Biomarkers <bioanalysisandbiomarkers.blogspot.com>
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